Аннотация:
Aza-Michael reaction of (E)-4-(diphenylphosphoryl)but-3-en-2-one with mono- and bicyclic nitrogen heterocycles proceeds regioselectively in the absence of catalysts to give the corresponding ß-diphenylphosphoryl-b-azahetarylalkanones. Its reaction with imidazole in the presence of chiral organocatalysts affords the corresponding enantiomerically enriched adduct in higher yield.
Тип публикации:
Статья
Язык публикации: английский
Образец цитирования:
M. A. Galkina, G. V. Bodrin, E. I. Goryunov, I. B. Goryunova, A. S. Sherstneva, J. S. Urmambetova, N. G. Kolotyrkina, M. M. Il'in, V. K. Brel, K. A. Kochetkov, “Regioselective aza-Michael addition of azoles to 4-(diphenylphosphoryl)but-3-en-2-one”, Mendeleev Commun., 26:1 (2016), 75–76
Образцы ссылок на эту страницу:
https://www.mathnet.ru/rus/mendc2116
https://www.mathnet.ru/rus/mendc/v26/i1/p75
Эта публикация цитируется в следующих 6 статьяx:
Alexander Yu. Rulev, “Weak Nucleophiles in the Aza‐Michael Reaction”, Adv Synth Catal, 365:12 (2023), 1908
Charanjit Kaur, Sachin Sharma, Amandeep Thakur, Ram Sharma, “Asymmetric Synthesis: A Glance at Various Methodologies for Different Frameworks”, COC, 26:8 (2022), 771
Zheng Li, Aizhen Yang, Xiaolong Ma, Zhenrong Liu, “Chemoselective aza-Michael addition of indoles to 2-aroyl-1,3-diarylenones”, Journal of Chemical Research, 44:1-2 (2020), 97
Maxim G. Vinogradov, Olga V. Turova, Sergei G. Zlotin, “Recent advances in the asymmetric synthesis of pharmacology-relevant nitrogen heterocyclesviastereoselective aza-Michael reactions”, Org. Biomol. Chem., 17:15 (2019), 3670
Maria A. Galkina, Georgy V. Bodrin, Evgenii I. Goryunov, Irina B. Goryunova, Aleksandra S. Sherstneva, Jumakan S. Urmambetova, Natalia G. Kolotyrkina, Mikhail M. Il'in, Valery K. Brel, Konstantin A. Kochetkov, “ChemInform Abstract: Regioselective Aza‐Michael Addition of Azoles to 4‐(Diphenylphosphoryl)but‐3‐en‐2‐one.”, ChemInform, 47:24 (2016)
Georgy V. Bodrin, Anna G. Matveeva, Evgenii I. Goryunov, Margarita P. Pasechnik, Rinat R. Aysin, Alexander N. Turanov, Vasilii K. Karandashev, Evgeny D. Savin, Alexander S. Peregudov, Yulia V. Nelyubina, Valery K. Brel, “The synthesis and extraction properties of new 2-(phosphorylalkyl)-and 2-(phosphorylalkenyl)-substituted 1,8- and 1,6-naphthyridines”, Chem Heterocycl Comp, 52:8 (2016), 583
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