Аннотация:
A series of new furazan (1,2,5-oxadiazole) derivatives based on structural overlap with combretastatin have been synthesized. Targeted molecules were evaluated using the sea urchin embryo assay; several agents demonstrated 1–4μmol dm–3 antiproliferative activity in this in vivo model.
Образец цитирования:
A. B. Sheremetev, D. E. Dmitriev, N. K. Lagutina, M. M. Raikhshtat, A. S. Kiselev, M. N. Semenova, N. N. Ikizalp, V. V. Semenov, “New functionalized aminofurazans as potential antimitotic agents in the sea urchin embryo assay”, Mendeleev Commun., 20:3 (2010), 132–134
Образцы ссылок на эту страницу:
https://www.mathnet.ru/rus/mendc3013
https://www.mathnet.ru/rus/mendc/v20/i3/p132
Эта публикация цитируется в следующих 12 статьяx:
Gülşah KURT, Fatih SEVGİ, “Synthesis and Biological Evaluation of Imidazole-2-thione Fused Furazan as a New Biheterocyclic Scaffold”, Düzce Üniversitesi Bilim ve Teknoloji Dergisi, 10:1 (2022), 14
E. B. Rakhimova, V. Yu. Kirsanov, E. S. Meshcheryakova, L. U. Dzhemileva, V. A. D'yakonov, A. G. Ibragimov, U. M. Dzhemilev, “Synthesis and cytotoxic activity of new annulated furazan derivatives”, Mendeleev Commun., 31:3 (2021), 362–364
Fedor E. Teslenko, Artem I. Churakov, Alexander A. Larin, Ivan V. Ananyev, Leonid L. Fershtat, Nina N. Makhova, “Route to 1,2,4- and 1,2,5-oxadiazole ring assemblies via a one-pot condensation/oxidation protocol”, Tetrahedron Letters, 61:13 (2020), 151678
Leire Mijangos, Martin Krauss, Laura de Miguel, Haizea Ziarrusta, Maitane Olivares, Olatz Zuloaga, Urtzi Izagirre, Tobias Schulze, Werner Brack, Ailette Prieto, Nestor Etxebarria, “Application of the Sea Urchin Embryo Test in Toxicity Evaluation and Effect-Directed Analysis of Wastewater Treatment Plant Effluents”, Environ. Sci. Technol., 54:14 (2020), 8890
Н. Н. Махова, Л. И. Беленький, Г. А. Газиева, И. Л. Далингер, Л. С. Константинова, В. В. Кузнецов, А. Н. Кравченко, М. М. Краюшкин, О. А. Ракитин, А. М. Старосотников, Л. Л. Ферштат, С. А. Шевелев, В. З. Ширинян, В. Н. Яровенко, “Прогресс в химии азот-, кислород- и серасодержащих гетероциклических систем”, Усп. хим., 89:1 (2020), 55–124; N. N. Makhova, L. I. Belen'kii, G. A. Gazieva, I. L. Dalinger, L. S. Konstantinova, V. V. Kuznetsov, A. N. Kravchenko, M. M. Krayushkin, O. A. Rakitin, A. M. Starosotnikov, L. L. Fershtat, S. A. Shevelev, V. Z. Shirinian, V. N. Yarovenko, “Progress in the chemistry of nitrogen-, oxygen- and sulfur-containing heterocyclic systems”, Russian Chem. Reviews, 89:1 (2020), 55–124
Elena B. Rakhimova, Victor Yu. Kirsanov, Ekaterina S. Mescheryakova, Leonard M. Khalilov, Askhat G. Ibragimov, Lilya U. Dzhemileva, Vladimir A. D'yakonov, Usein M. Dzhemilev, “First Example of Catalytic Synthesis of Difurazanohexahydrohexaazapyrenes and in Vitro Study of Their Antitumor Activity”, ACS Med. Chem. Lett., 10:3 (2019), 378
Andrei I. Stepanov, Dmitry V. Dashko, Elena V. Stepanova, “3-Amino-4-[5-(chloromethyl)-1,2,4-oxadiazol-3-yl]furazan –a multifunctional synthon for the synthesis of 1,2,5-oxadiazole derivatives”, Chem Heterocycl Comp, 55:12 (2019), 1233
Andrei I. Stepanov, Alexander A. Astrat'ev, Aleksei B. Sheremetev, Nataliya K. Lagutina, Nadezhda V. Palysaeva, Aleksei Yu. Tyurin, Nataliya S. Aleksandrova, Nataliya P. Sadchikova, Kyrill Yu. Suponitsky, Olga P. Atamanenko, Leonid D. Konyushkin, Roman V. Semenov, Sergei I. Firgang, Alex S. Kiselyov, Marina N. Semenova, Victor V. Semenov, “A facile synthesis and microtubule-destabilizing properties of 4-(1H-benzo[d]imidazol-2-yl)-furazan-3-amines”, European Journal of Medicinal Chemistry, 94 (2015), 237
D. E. Dmitriev, Yu. A. Strelenko, A. B. Sheremetev, “NMR spectroscopic study of 3-nitrofurazans”, Russ Chem Bull, 62:2 (2013), 504
D. V. Tsyganov, N. B. Chernysheva, L. K. Salamandra, L. D. Konyushkin, O. P. Atamanenko, M. N. Semenova, V. V. Semenov, “Synthesis of Polyalkoxy-3-(4-Methoxyphenyl)Coumarins with Antimitotic Activity from Plant Allylpolyalkoxybenzenes”, Mendeleev Commun., 23:3 (2013), 147–149
Aleksei B. Sheremetev, Nadezhda V. Palysaeva, Marina I. Struchkova, Kyrill Yu. Suponitsky, Mikhail Yu. Antipin, “Copper‐Catalyzed C–N Coupling Reactions of Nitrogen‐Rich Compounds – Reaction of Iodofurazans with s‐Tetrazinylamines”, Eur J Org Chem, 2012:11 (2012), 2266
Aleksei B. Sheremetev, Dmitrii E. Dmitriev, Nataliya K. Lagutina, Mikhail M. Raihstat, Alex S. Kiselyov, Marina N. Semenova, Natalie N. Ikizalp, Victor V. Semenov, “ChemInform Abstract: New Functionalized Aminofurazans as Potential Antimitotic Agents in the Sea Urchin Embryo Assay.”, ChemInform, 41:45 (2010)
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