Аннотация:
Reaction of thiosemicarbazide with carboxylic acids, including N-substituted amino acids, in ionic liquids with H2SO4 as a catalyst affords 5-R-2-amino-1,3,4-thiadiazoles. On using alkanedicarboxylic acids, α,ω-bis(2-amino-1,3,4,-thiadiazol-5-yl)alkanes were obtained.
Образец цитирования:
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Nguyen Dinh Thanh, Vu Ngoc Toan, Nguyen Thi Kim Giang, Hoang Thi Kim Van, Do Son Hai, Nguyen Minh Tri, Duong Ngoc Toan, “Synthesis, biological and molecular modelling for 1,3,4-thiadiazole sulfonyl thioureas: bacterial and fungal activity”, RSC Med. Chem., 14:12 (2023), 2751
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Arti Vishwkarma, A.K. Srivastava, O.P. Pandey, S.K. Sengupta, “Zinc(II) Complexes of Schiff Bases Derived from Bis-(2-hydrazino-1,3,4-thiadiazole-5-
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M. A. Epishina, A. S. Kulikov, N. V. Ignat'ev, M. Schulte, N. N. Makhova, “Efficient synthesis of tertiary acyclic amides by the Chapman rearrangement of aryl benzimidates in ionic liquids”, Mendeleev Commun., 25:2 (2015), 126–128
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N. N. Makhova, M. I. Pleshchev, M. A. Epishina, A. S. Kulikov, “Synthesis and Transformations of Nitrogen Heterocycles in Ionic Liquids (Review)”, Chem Heterocycl Comp, 50:5 (2014), 634
Margarita A. Epishina, Alexander S. Kulikov, Nikolai V. Ignat'ev, Michael Schulte, Nina N. Makhova, “ChemInform Abstract: Synthesis of 5‐Alkyl‐2‐amino‐1,3,4‐thiadiazoles and α,ω‐Bis(2‐amino‐1,3,4‐thiadiazol‐5‐yl)alkanes in Ionic Liquids.”, ChemInform, 43:17 (2012)
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