Abstract:
Two six-step syntheses of 6-acetylamino(indolo[2,3-b])bicyclo[3.2.1]oct-2-ene 2 and 6-acetylamino(5’-methoxyindolo[2,3-b])-bicyclo[3.2.1]oct-2-ene 3 are presented, and the crystal structure of compound 2 is described.
Citation:
T. Yu. Baranova, N. V. Averina, N. V. Zyk, N. S. Zefirov, K. A. Lyssenko, M. Yu. Antipin, O. N. Zefirova, “Synthesis of indole derivatives fused with bicyclo[3.2.1]octane framework”, Mendeleev Commun., 19:1 (2009), 10–11
Linking options:
https://www.mathnet.ru/eng/mendc3099
https://www.mathnet.ru/eng/mendc/v19/i1/p10
This publication is cited in the following 6 articles:
I. B. Davydova, V. M. Senyavin, O. N. Zefirova, G. M. Kuramshina, “Vibrational Spectra and Stable Conformations of (1RS, 5RS, 6SR)-6-Methoxycarbonylamino-(5'-methoxyindolo[2,3-b])bicyclo[3.2.1]oct-2-en”, Russ. J. Phys. Chem., 93:8 (2019), 1525
D. V. Shishov, E. V. Nurieva, N. S. Zefirov, A. V. Mamaeva, O. N. Zefirova, “Synthesis of 5-hydroxy-4-methoxytricyclo[7.3.1.02,7]trideca-2,4,6-trien- 8-one – precursor of putative bioisosteric colchicine analogues”, Mendeleev Commun., 24:6 (2014), 370–371
T. Yu. Baranova, O. N. Zefirova, A. M. Banaru, V. N. Khrustalev, A. A. Ivanova, A. A. Ivanov, N. S. Zefirov, “Crystallographic study and molecular modeling on the oxidation product of N-[(8R)-2-methoxy-5,6,7,8,9,10-hexahydro-6,9-methanocyclohepta[b]indol-8-yl]acetamide”, Russ J Org Chem, 48:4 (2012), 552
O. N. Zefirova, T. Yu. Baranova, K. A. Lyssenko, N. A. Zefirov, N. V. Zyk, P. M. Vassiliev, D. S. Yakovlev, A. A. Spasov, “Synthesis and biological testing of conformationally restricted serotonin analogues with bridgehead moieties”, Mendeleev Commun., 22:2 (2012), 75–77
Olga N. Zefirova, Tatiana Yu Baranova, Anna A. Ivanova, Andrei A. Ivanov, Nikolay S. Zefirov, “Application of the bridgehead fragments for the design of conformationally restricted melatonin analogues”, Bioorganic Chemistry, 39:2 (2011), 67
Tatiana Yu. Baranova, Nadezhda V. Averina, Nikolai V. Zyk, Nikolai S. Zefirov, Konstantin A. Lyssenko, Mikhail Yu. Antipin, Olga N. Zefirova, “ChemInform Abstract: Synthesis of Indole Derivatives Fused with Bicyclo[3.2.1]octane Framework.”, ChemInform, 40:29 (2009)